高效,快速,以及高收率的芳基席夫碱衍生物的合成及其对 hCA I 的体外和硅抑制研究 ,HCA II,AChE,还有 BuChe.
关键词: 1,2,4‐triazole Alzheimer's disease Schiff base carbonic anhydrase cholinesterase
Mesh : Schiff Bases / pharmacology chemistry chemical synthesis Cholinesterase Inhibitors / pharmacology chemical synthesis chemistry Butyrylcholinesterase / metabolism Acetylcholinesterase / metabolism Humans Carbonic Anhydrase II / antagonists & inhibitors metabolism Carbonic Anhydrase Inhibitors / pharmacology chemical synthesis chemistry Carbonic Anhydrase I / antagonists & inhibitors metabolism Structure-Activity Relationship Molecular Structure Molecular Docking Simulation Computer Simulation Dose-Response Relationship, Drug Models, Molecular
来 源: DOI:10.1002/ardp.202300266