%0 Journal Article %T Synthesis and biological evaluation of acylthiourea against DUSP1 inhibition. %A Yeon Kim B %A Hee Yoon J %A Kim M %A Nyoung Kim J %A Park H %A Eon Ryu S %A Lee S %J Bioorg Med Chem Lett %V 29 %N 14 %D 07 2019 15 %M 31103445 %F 2.94 %R 10.1016/j.bmcl.2019.05.021 %X Structure based virtual screening attempts to discover DUSP1 inhibitors have yielded a scaffold featuring benzoxazole and acylthiourea pharmacophore. A series of its analogues were synthesized to explore structure activity relationship (SAR) of DUSP1 inhibition.