%0 Journal Article %T Thermodynamic optimisation in drug discovery: a case study using carbonic anhydrase inhibitors. %A Scott AD %A Phillips C %A Alex A %A Flocco M %A Bent A %A Randall A %A O'Brien R %A Damian L %A Jones LH %J ChemMedChem %V 4 %N 12 %D Dec 2009 %M 19882701 %F 3.54 %R 10.1002/cmdc.200900386 %X